平安! 发表于 2011-11-9 19:57
t+ d6 J; W3 nPazopanib (100 mg/kg/day free base equivalent) # S0 ]2 R9 q% L Z5 b
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。$ v. N( j# _" |8 o4 x/ _ W
搜索了一下,原料一大堆。
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/ S6 |1 \7 C8 ~# [, w. B对不起!100mg/kg是用于移植瘤的,我弄错了。
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* W0 U- u; V3 D- ]. t0 v以下是正版说明书的推荐用量。. b) R( n! U: H7 k0 L
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--------------------- DOSAGE AND ADMINISTRATION ----------------
% i' [; F; P& j* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) ) l( U& p6 H/ `" n6 f
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) " u% ?5 o9 L: d4 o T1 v
---------------------DOSAGE FORMS AND STRENGTHS --------------
' y$ U- k( ] V5 L# I- k200 mg tablets. (3)
8 n3 Q: m/ d/ T-------------------------------CONTRAINDICATIONS------------------------ |