平安! 发表于 2011-11-9 19:57
" o4 ~! H. t$ g* W: i* UPazopanib (100 mg/kg/day free base equivalent) * }$ }0 p( \' x" V' @
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。- y3 u, w( p3 h# L$ p. |! G5 D1 A* r& ]
搜索了一下,原料一大堆。
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对不起!100mg/kg是用于移植瘤的,我弄错了。
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以下是正版说明书的推荐用量。
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--------------------- DOSAGE AND ADMINISTRATION ----------------+ k0 q! V& [6 @5 e' _% W6 C+ k
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
# y7 p+ v% ^. K+ j* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
# ^# ^# d a* j: d% U, n---------------------DOSAGE FORMS AND STRENGTHS --------------
$ T! F4 t y# U200 mg tablets. (3)
8 ?( k8 B1 I' i5 H b: {( v8 ^0 P+ G# M-------------------------------CONTRAINDICATIONS------------------------ |